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Afatinib (BIBW2992) Dimaleate [850140-73-7]

Research Use Only
S7810
Selleck Chemicals
Product group Chemicals
Price on request
Packing Size
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Afatinib (BIBW2992) Dimaleate [850140-73-7]
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Scientific Description
    Afatinib (BIBW2992) Dimaleate irreversibly inhibits EGFR/HER2 including EGFR(wt), EGFR(L858R), EGFR(L858R/T790M) and HER2 with IC50 of 0.5 nM, 0.4 nM, 10 nM and 14 nM, respectively; 100-fold more active against Gefitinib-resistant L858R-T790M EGFR mutant. Afatinib (BIBW2992) Dimaleate induces autophagy.
  • UNSPSC
    12352200