Sapitinib (AZD8931) [848942-61-0]
S2192
Overview
- SupplierSelleck Chemicals
- Product NameSapitinib (AZD8931) [848942-61-0]
- Delivery Days Customer9
- CAS Number848942-61-0
- CertificationResearch Use Only
- Scientific DescriptionSapitinib (AZD8931) is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4 nM, 3 nM and 4 nM in cell-free assays, more potent than Gefitinib or Lapatinib against NSCLC cell, 100-fold more selective for the ErbB family than MNK1 and Flt. Phase 2.
- UNSPSC12352200