Baclofen [1134-47-0]

MedChem Express

Baclofen [1134-47-0]

10

1134-47-0

99.42%

C10H12ClNO2

213.66

Baclofen, a lipophilic derivative of gamma-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research.

O=C(O)CC(C1=CC=C(Cl)C=C1)CN

2°C to 8°C,-20°C,-80°C

12352200