Pinometostat (EPZ5676) [1380288-87-8]
S7062
Product group Chemicals
Overview
- SupplierSelleck Chemicals
- Product NamePinometostat (EPZ5676) [1380288-87-8]
- Delivery Days Customer9
- CertificationResearch Use Only
- Scientific DescriptionPinometostat (EPZ5676) is an S-adenosyl methionine (SAM) competitive inhibitor of protein methyltransferase DOT1L with Ki of 80 pM in a cell-free assay, demonstrating >37,000-fold selectivity against all other PMTs tested, inhibits H3K79 methylation in tumor. Phase 1.
- UNSPSC12352200