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Imidafenacin [170105-16-5]

Research Use Only
S5385
Selleck Chemicals
CAS Number170105-16-5
Product group Chemicals
Price on request
Packing Size
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Imidafenacin [170105-16-5]
  • Delivery Days Customer
    9
  • CAS Number
    170105-16-5
  • Certification
    Research Use Only
  • Scientific Description
    Imidafenacin (KRP-197, ONO-8025) is a urinary antispasmodic of the anticholinergic class. It is a novel antimuscarinic agent with safety and efficacy, has been clinically used for the treatment of overactive bladder. Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). IC50 value: 0.3 nM(M3).
  • UNSPSC
    12352200