Netupitant [290297-26-6]

MedChem Express

Netupitant [290297-26-6]

10

290297-26-6

98.96%

C30H32F6N4O

578.59

Netupitant (CID-6451149) is a highly potent, selective and orally active neurokinin-1 (NK1) receptor antagonist with a Ki of 0.95 nM for hNK1 in CHO cells. Netupitant has antiemetic affect.

CN1CCN(C2=CC(C3=C(C)C=CC=C3)=C(N(C)C(C(C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)(C)C)=O)C=N2)CC1

2°C to 8°C,-20°C,-80°C

12352200