Olcegepant hydrochloride [586368-06-1]

MedChem Express

Olcegepant hydrochloride [586368-06-1]

10

586368-06-1

Research Use Only

99.11%

C38H47Br2N9O5.HCl

906.11

Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.

O=C1N(CC2=C(N1)C=CC=C2)C3CCN(C(N[C@@H](C(N[C@H](C(N4CCN(C5=CC=NC=C5)CC4)=O)CCCCN)=O)CC6=CC(Br)=C(C(Br)=C6)O)=O)CC3.Cl

2°C to 8°C,-20°C,-80°C

12352200