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Birabresib (OTX015) [202590-98-5]

Research Use Only
S7360
Selleck Chemicals
CAS Number202590-98-5
Product group Chemicals
Price on request
Packing Size
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Birabresib (OTX015) [202590-98-5]
  • Delivery Days Customer
    9
  • CAS Number
    202590-98-5
  • Certification
    Research Use Only
  • Scientific Description
    Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
  • UNSPSC
    12352200