Bio-Connect

PKC-IN-1 [1046787-18-1]

HY-16903
MedChem Express
CAS Number1046787-18-1
Product group Chemicals
Estimated Purity98.79%
Molecular Weight500.61
Price on request
Packing Size
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    PKC-IN-1 [1046787-18-1]
  • Delivery Days Customer
    10
  • CAS Number
    1046787-18-1
  • Estimated Purity
    98.79%
  • Molecular Formula
    C25H37FN8O2
  • Molecular Weight
    500.61
  • Scientific Description
    PKC-IN-1 is a potent, ATP-competitive and reversible inhibitor of conventional PKC enzymes with Kis of 5.3 and 10.4 nM for human PKCbeta and PKCalpha, and IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM for PKCalpha, PKCbetaI, PKCbetaII, PKCtheta, PKCgamma, PKC mu and PKCepsilon, respectively.
  • SMILES
    O=C(N1[C@@H](C)CN(CC2CCOCC2)[C@H](C)C1)N(C3)C(C)(C)C4=C3C(NC5=NC(C)=NC=C5F)=NN4
  • Storage Instruction
    2°C to 8°C,-20°C,-80°C
  • UNSPSC
    12352200