PROTAC ERalpha Degrader-2 [1351169-29-3]

MedChem Express

PROTAC ERalpha Degrader-2 [1351169-29-3]

10

1351169-29-3

98.02%

C42H61N5O8

763.96

PROTAC ERalpha Degrader-2 comprises a IAP ligand binding group, a linker and an estrogen receptor alpha (ERalpha) binding group. PROTAC ERalpha Degrader-2 is an ERalpha degrader. Maximal ERalpha degradation at 30 microM concentration in human mammary tumor MCF7 cells. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs).

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-20°C,-80°C

12352200