Setipiprant [866460-33-5]
HY-16635
Overview
- SupplierMedChem Express
- Product NameSetipiprant [866460-33-5]
- Delivery Days Customer10
- CAS Number866460-33-5
- CertificationResearch Use Only
- Estimated Purity98.7%
- Molecular FormulaC24H19FN2O3
- Molecular Weight402.42
- Scientific DescriptionSetipiprant (ACT-129968) is an orally active and selective CRTH2 antagonist. Setipiprant interacts with hCRTH2 receptor with an IC50 value of 6 nM. Setipiprant inhibits prostanoid receptors hDP1 and hEP2 with IC50 values of 1290 and 2600 nM, respectively. Setipiprant can be used for the research of asthma and rhinitis.
- SMILESO=C(O)CN1C2=C(CN(C(C3=C4C=CC=CC4=CC=C3)=O)CC2)C5=C1C=CC(F)=C5
- Storage Instruction2°C to 8°C,-20°C,-80°C
- UNSPSC12352200