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Tivantinib (ARQ 197) [905854-02-6]

Research Use Only
S2753
Selleck Chemicals
CAS Number905854-02-6
Product group Chemicals
Price on request
Packing Size
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Tivantinib (ARQ 197) [905854-02-6]
  • Delivery Days Customer
    9
  • CAS Number
    905854-02-6
  • Certification
    Research Use Only
  • Scientific Description
    Tivantinib (ARQ 197) is the first non-ATP-competitive c-Met inhibitor with Ki of 0.355 muM in a cell-free assay, little activity to Ron, and no inhibition to EGFR, InsR, PDGFRalfa or FGFR1/4. Tivantinib (ARQ 197) induces a G2/M arrest and apoptosis. Phase 3.
  • UNSPSC
    12352200