WH-4-023 [837422-57-8]
S7565
Overview
- SupplierSelleck Chemicals
- Product NameWH-4-023 [837422-57-8]
- Delivery Days Customer9
- CAS Number837422-57-8
- CertificationResearch Use Only
- Scientific DescriptionWH-4-023 (KIN001-112, KIN112, Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor with IC50s of 2 nM and 6 nM in cell-free assays, respectively. Exhibits >300-fold selectivity against p38alfa and KDR. Also potently inhibits SIK (IC50 values are 10, 22 and 60 nM for SIK 1, 2 and 3 respectively) and displays selectivity over a range of closely related kinases.
- UNSPSC12352200