Fulvestrant [129453-61-8]

MedChem Express

Fulvestrant [129453-61-8]

10

129453-61-8

Research Use Only

95%

C32H47F5O3S

606.77

Fulvestrant (ICI 182780) is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC50 of 9.4 nM. Fulvestrant is also a GPR30 agonist. Fulvestrant effectively inhibits the growth of ER-positive MCF-7 cells with an IC50 of 0.29 nM. Fulvestrant also induces autophagy and has antitumor efficacy.

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2°C to 8°C,-20°C,-80°C

12352200