LP-211 [1052147-86-0]

Biorbyt

LP-211 [1052147-86-0]

16

1052147-86-0

Research Use Only

C28N3O5CL2H23

552.4053

LP-211 is a selective and blood-brain barrier penetrant 5-HT7 receptor agonist, with a Ki of 0.58 nM, with high selectivity over 5-HT1A receptor (Ki, 188 nM) and D2 receptor (Ki, 142 nM).

ClC1C([H])=C([H])C([H])=C(C=1C1C(C([H])([H])OC2C([H])=C([H])C(=C([H])C=2[H])C2(C([H])([H])N(C3C([H])=C(C(=O)O[H])C([H])=C([H])N=3)C2([H])[H])O[H])=C(C2([H])C([H])([H])C2([H])[H])ON=1)Cl

12352200