Tasimelteon [609799-22-6]
S4281
Overview
- SupplierSelleck Chemicals
- Product NameTasimelteon [609799-22-6]
- Delivery Days Customer9
- CAS Number609799-22-6
- CertificationResearch Use Only
- Scientific DescriptionTasimelteon (BMS 214778, VEC 162) is a selective dual melatonin receptor (MT1/MT2) agonist with 2.1-4.4 times greater affinity for the MT2 receptor believed to mediate circadian rhythm phase-shifting (Ki = 0.0692 nM and Ki = 0.17 nM in NIH-3T3 and CHOeK1 cells, respectively), than for the MT1 receptor (Ki = 0.304 nM and Ki = 0.35 nM, respectively).
- UNSPSC12352200